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Found 27 from Tel-Aviv University
TargetReverse transcriptase(Human immunodeficiency virus 1)
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50478430(CHEMBL500695)
Affinity DataIC50:  24nMAssay Description:Inhibition of HIV1 reverse transcriptase activity assessed as residual enzyme activity by poly(rA)n.oligo(dT)12-18-directed incorporation of [3H]dTTP...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50478436(CHEMBL448380)
Affinity DataIC50:  77nMAssay Description:Inhibition of HIV1 reverse transcriptase activity assessed as residual enzyme activity by poly(rA)n.oligo(dT)12-18-directed incorporation of [3H]dTTP...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50478431(CHEMBL455390)
Affinity DataIC50:  112nMAssay Description:Inhibition of HIV1 reverse transcriptase activity assessed as residual enzyme activity by poly(rA)n.oligo(dT)12-18-directed incorporation of [3H]dTTP...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50491950(CHEMBL2386692)
Affinity DataIC50:  821nMAssay Description:Inhibition of trypsin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50491950(CHEMBL2386692)
Affinity DataIC50:  821nMAssay Description:Inhibition of trypsin (unknown origin) using benzoyl-L-arginine-p-nitroanilide hydrochloride as substrate preincubated for 5 mins before substrate ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) antiporter NhaA(Escherichia coli (strain K12))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50010751(1H,3H-Perimidin-2-ylideneamine | 2-aminoperimidine...)
Affinity DataIC50:  1.70E+3nMAssay Description:Antiporter activity in Escherichia coli K12 wild type EcNhaA assessed as effect on sodium chloride-induced pH changes by acridine orange fluorescence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) antiporter NhaA(Escherichia coli (strain K12))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50010751(1H,3H-Perimidin-2-ylideneamine | 2-aminoperimidine...)
Affinity DataIC50:  2.20E+3nMAssay Description:Antiporter activity in Escherichia coli K12 wild type EcNhaA assessed as effect on lithium chloride-induced pH changes by acridine orange fluorescenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50491951(CHEMBL2386691)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of trypsin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50478437(CHEMBL506716)
Affinity DataIC50:  2.95E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase activity assessed as residual enzyme activity by poly(rA)n.oligo(dT)12-18-directed incorporation of [3H]dTTP...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50491948(CHEMBL2386693)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of trypsin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50491949(CHEMBL2386694)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of trypsin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50494500(CHEMBL3092720)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of trypsin (unknown origin) using benzoyl-L-arginine-p-nitroanilide hydrochloride as substrate preincubated for 5 mins before substrate ad...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50494501(CHEMBL3092721)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of trypsin (unknown origin) using benzoyl-L-arginine-p-nitroanilide hydrochloride as substrate preincubated for 5 mins before substrate ad...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50494503(CHEMBL3092723)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of thrombin (unknown origin) using z-Gly-Pro-Arg-4MbetaNA-acetate as substrate preincubated for 20 mins before substrate addition measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50494502(CHEMBL3092722)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of trypsin (unknown origin) using benzoyl-L-arginine-p-nitroanilide hydrochloride as substrate preincubated for 5 mins before substrate ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50494503(CHEMBL3092723)
Affinity DataIC50:  3.08E+4nMAssay Description:Inhibition of trypsin (unknown origin) using benzoyl-L-arginine-p-nitroanilide hydrochloride as substrate preincubated for 5 mins before substrate ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50478432(CHEMBL448268)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase activity assessed as residual enzyme activity by poly(rA)n.oligo(dT)12-18-directed incorporation of [3H]dTTP...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50312534(CHEMBL1076839 | cyanopeptolin SS)
Affinity DataIC50:  4.52E+4nMAssay Description:Inhibition of thrombin after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50491918(CHEMBL2011690)
Affinity DataIC50:  4.55E+4nMAssay Description:Inhibition of trypsin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50312533((R)-N-((2S,5S,8S,11R,12S,15S,18S,21R)-5-benzyl-2,8...)
Affinity DataIC50:  5.29E+4nMAssay Description:Inhibition of thrombin after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50478438(CHEBI:90507 | CHEMBL499250)
Affinity DataIC50:  6.50E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase activity assessed as residual enzyme activity by poly(rA)n.oligo(dT)12-18-directed incorporation of [3H]dTTP...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50478434(CHEMBL470759)
Affinity DataIC50:  7.50E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase activity assessed as residual enzyme activity by poly(rA)n.oligo(dT)12-18-directed incorporation of [3H]dTTP...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50478433(CHEMBL447743)
Affinity DataIC50:  9.94E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase activity assessed as residual enzyme activity by poly(rA)n.oligo(dT)12-18-directed incorporation of [3H]dTTP...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50478440(CHEMBL472021)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HIV1 reverse transcriptase activity assessed as residual enzyme activity by poly(rA)n.oligo(dT)12-18-directed incorporation of [3H]dTTP...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50478439(CHEBI:63774 | CHEMBL443117)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HIV1 reverse transcriptase activity assessed as residual enzyme activity by poly(rA)n.oligo(dT)12-18-directed incorporation of [3H]dTTP...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50478435(CHEMBL450754)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HIV1 reverse transcriptase activity assessed as residual enzyme activity by poly(rA)n.oligo(dT)12-18-directed incorporation of [3H]dTTP...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Tel-Aviv University

Curated by ChEMBL
LigandPNGBDBM50478441(CHEBI:15754 | CHEMBL446492)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HIV1 reverse transcriptase activity assessed as residual enzyme activity by poly(rA)n.oligo(dT)12-18-directed incorporation of [3H]dTTP...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed